Antibodies
(R)-baclofen
- 貨號 Cat. No.
- S3072
- 規格 Size
- 10mgã€50mg
- 品牌 Brand
- Selleckchem
Description
(R)-baclofen
Catalog No.S3072
(R)-baclofen is a derivative of gamma-aminobutyric acid primarily used to treat spasticity.
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Biological Activity
| Description | (R)-baclofen is a derivative of gamma-aminobutyric acid primarily used to treat spasticity. | |||||
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| Targets | ||||||
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| In vitro | Baclofen is a skeletal muscle relaxant used in the treatment of spasticity of spinal and cerebral origin. Although it is marketed as a racemic mixture, only the baclofen R-enantiomer is stereospecifically active at so called GAGAB-receptors. [1] Researchers believe that the enantiomers of baclofen have different properties. It is claimed that the R-(−)-enantiomer is about 100 times more active than the S-(+)-enantiomer. | |||||
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| Features | ||||||
Protocol(Only for Reference)
References
Chemical Information
| Molecular Weight (MW) | 213.66 |
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| Formula | C10H12ClNO2 |
| CAS No. | 69308-37-8 |
| Storage | 3 years -20℃Powder |
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| 6 months-80℃in DMSO | |
| Syonnyms | N/A |
| Solubility (25°C) * | In vitro | DMSO | <1 mg/mL (<1 mM) |
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| Water | 8 mg/mL (37 mM) | ||
| Ethanol | <1 mg/mL (<1 mM) | ||
| * <1 mg/ml means slightly soluble or insoluble. * Please note that Selleck tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. | |||
| Chemical Name | Benzenepropanoic acid, β-(aminomethyl)-4-chloro-, (βR)- |
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