PHA-739358
Chemical Compounds
- 貨號 Cat. No.
- M1769
- 規格 Size
- 10mg,50mg
- 品牌 Brand
- No Brand
Description
PHA-739358 (Danusertib) is a small molecule with low nanomolar activity against all aurora kinases (AKs) with IC50 value of 13 nM for aurora-A and 79 nM for aurora-B respectively. PHA-739358 (Danusertib) also inhibits other cancer relevant tyrosine kinases such as wild type and mutated ABL, RET, TRK-A and FGFRs.

