PHA-739358

Chemical Compounds

貨號 Cat. No.
M1769
規格 Size
10mg,50mg
品牌 Brand
No Brand

Description

PHA-739358 (Danusertib) is a small molecule with low nanomolar activity against all aurora kinases (AKs) with IC50 value of 13 nM for aurora-A and 79 nM for aurora-B respectively. PHA-739358 (Danusertib) also inhibits other cancer relevant tyrosine kinases such as wild type and mutated ABL, RET, TRK-A and FGFRs.

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