Antibodies
Gabapentin
- 貨號 Cat. No.
- S2133
- 規格 Size
- 25mgã€100mg
- 品牌 Brand
- Selleckchem
Description
GabapentinLicensed by Pfizer
Catalog No.S2133
Gabapentin is a pharmaceutical agent, specifically a GABA analogue.
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Distributor Tel: +886-2-2827-1197jimmy@new.abscience.com.tw
Biological Activity
Gabapentin (Neurontin) is a pharmaceutical agent, specifically a GABA analogue. Gabapentin (Neurontin) was originally developed for the treatment of epilepsy, and currently, gabapentin is widely used to relieve pain, especially neuropathic pain. Its therapeutic action on neuropathic pain is thought to involve voltage-gated N-type calcium ion channels. It is thought to bind to the α2δ subunit (1 and 2) of the voltage-dependent calcium channel in the central nervous system. [1][2]
Clinical Trial Information( data from http://clinicaltrials.gov)
| NCT Number | Recruitment | Conditions | Sponsor /Collaborators | Start Date | Phases |
|---|---|---|---|---|---|
| NCT02127853 | Not yet recruiting | Hyperalgesia | Seoul National University Hospital | Phase 4 | |
| NCT02117076 | Recruiting | Restless Leg Syndrome | University of South Florida|Theresa Zesiewicz|Lehigh Valley Hospital | Phase 4 | |
| NCT02064790 | Enrolling by invitation | Radicular; Neuropathic, Lumbar, Lumbosacral|Radicular; Neuropathic, Cervical | Emory University | ||
| NCT01852318 | Not yet recruiting | Uremic Pruritus | National Taiwan University Hospital|Cathay General Hospital | Phase 4 | |
| NCT02076893 | Recruiting | Pain | Children’s Hospitals and Clinics of Minnesota | Phase 4 |
Chemical Information
| Molecular Weight (MW) | 171.24 |
|---|---|
| Formula | C9H17NO2 |
| CAS No. | 60142-96-3 |
| Storage | 3 years -20℃Powder |
|---|---|
| 6 months-80℃in DMSO | |
| Syonnyms | Fanatrex, Gabarone |
| Solubility (25°C) * | In vitro | DMSO | <1 mg/mL (<1 mM) |
|---|---|---|---|
| Water | 34 mg/mL (198 mM) | ||
| Ethanol | <1 mg/mL (<1 mM) | ||
| * <1 mg/ml means slightly soluble or insoluble. * Please note that Selleck tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. | |||
| Chemical Name | 2-(1-(aminomethyl)cyclohexyl)acetic acid |
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